Hepatic enzymatic transformation of drugs. Phase I (oxidation by CYP450) + phase II (conjugation by UGT, SULT). CYP3A4 metabolises ~50% of drugs. Drug-drug interactions via induction/inhibition.
Hepatic enzymatic transformation of drugs. Phase I (oxidation by CYP450) + phase II (conjugation by UGT, SULT). CYP3A4 metabolises ~50% of drugs. Drug-drug interactions via induction/inhibition.