Largest receptor family (~800 in humans): 7-transmembrane-helix receptors coupling ligand binding to heterotrimeric Gα/β/γ activation. Targets ~35% of FDA-approved drugs.
Largest receptor family (~800 in humans): 7-transmembrane-helix receptors coupling ligand binding to heterotrimeric Gα/β/γ activation. Targets ~35% of FDA-approved drugs.