T Blundell 1980s + Wlodawer HIV-protease 1989: X-ray structure-guided inhibitor design; saquinavir 1995 first SBDD-launched drug; modern fragment-based drug design.
T Blundell 1980s + Wlodawer HIV-protease 1989: X-ray structure-guided inhibitor design; saquinavir 1995 first SBDD-launched drug; modern fragment-based drug design.