Binding described by K_d = k_off/k_on; residence time t_res = 1/k_off increasingly recognised as better potency predictor than K_d alone. Competitive vs non-competitive vs allosteric modalities give distinct dose–response signatures.
Binding described by K_d = k_off/k_on; residence time t_res = 1/k_off increasingly recognised as better potency predictor than K_d alone. Competitive vs non-competitive vs allosteric modalities give distinct dose–response signatures.