Clark 1926: drug effect proportional to receptor occupancy. Agonist (activates), partial agonist (submax), antagonist (blocks), inverse agonist (reduces constitutive activity), allosteric modulator. Black Nobel 1988.
Clark 1926: drug effect proportional to receptor occupancy. Agonist (activates), partial agonist (submax), antagonist (blocks), inverse agonist (reduces constitutive activity), allosteric modulator. Black Nobel 1988.